Diacetylnalorphine

Diacetylnalorphine
Names
IUPAC name
: [(4R,4aR,7S,7aR,12bS)-9-acetyloxy-3-prop-2-enyl-2,4,4a,7,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-7-yl] acetate
Identifiers
2748-74-5
3D model (Jmol) Interactive image
ChEMBL ChEMBL2106214
ChemSpider 16736941
PubChem 20055473
Properties
C23H25NO5
Molar mass 395.4 g/mol
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
Infobox references

Diacetylnalorphine (BAN) is an opioid drug described as an analgesic and antidote which was never marketed.[1] It is the 3,6-diacetyl ester of nalorphine, and therefore the heroin analogue of nalorphine. Diacetylnalorphine may behave as a prodrug to nalorphine, similarly to the cases of heroin (diacetylmorphine) to morphine and diacetyldihydromorphine to dihydromorphine.

See also

References

  1. C.R. Ganellin; David J. Triggle (21 November 1996). Dictionary of Pharmacological Agents. CRC Press. pp. 1395–. ISBN 978-0-412-46630-4.



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